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þ ̿ MPT0B640 ú ȿ
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ϴ μ 輭 ִ 6 ġ ȿ
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۸ ؼ ڣ
þƹ̿ 8 HSP90 Ѱ 2 HSP90 MPT0B640 ϴб μҿ ڷγ19 ̷ ȿ ִٴ Ȯߴٰ ִ.
ϴ μҿ ڷγ19 MPT0B640 ̷ Ư Ȯϱ IC50 , MPT0B640 0-150nM 50% ̷ ҽװ, 300-750nM ִ 90-95% ̷ ƴ. Vero E6 MPT0B640 ̷ ȿ ָ, 50% (IC50) 72ð 118.7nM 24.86nM Ȯεƴ.
̹ ֵ ϴ μ 24ð, 48ð, 72ð پ MPT0B640 100nM ִ 72ð ̷ Ȱ ȿ ƴ϶ ġ ʾҴ. , MPT0B640 100nM ġ ʰ COVID-19 ϴ ȿ ִ١ ߴ.
þƹ̿ ú 72ð IC50 0.72M ݸ, MPT0B640 0.12M̱ ú ̷ Ȱ 6 ̻ ϴٰ ߴ. ƿ ó MPT0B640 ڷγ19 ̷ ȿ δٴ ̱ FDA ڷγ19 ߰ IND غ ߿ ִٰ .
ؼ (junsoo@mdtoday.co.kr)
<ǰ ̴ ѹα ǥ Ƿ, ǰ Ź , >
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