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þ ̿ ׾ MPT0B640 ú񸣺 ȿ
ϴ μ 輭 ִ 6 ġ ȿ
Ϻ Ʈ Ȯ Է : 2020-09-11 17:33:45

۸޵ ؼ ڣ

þƹ̿ 8 HSP90 Ѱ 2 HSP90 MPT0B640 ϴб μҿ ڷγ19 ׹̷ ȿ ִٴ Ȯߴٰ ִ.

ϴ μҿ ڷγ19 MPT0B640 ׹̷ Ư Ȯϱ IC50 , MPT0B640 0-150nM 50% ̷ ҽװ, 300-750nM 󵵿 ִ 90-95% ̷ ƴ. Vero E6 MPT0B640 ׹̷ ȿ ָ, 50% (IC50) 72ð 118.7nM 24.86nM Ȯεƴ.

̹ ֵ ϴ μ 24ð, 48ð, 72ð پ 󵵿 MPT0B640 100nM ִ 72ð ׹̷ Ȱ ȿ ƴ϶ ġ ʾҴ. , MPT0B640 100nM ġ ʰ COVID-19 ϴ ȿ ִ١ ߴ.

þƹ̿ ú񸣰 72ð IC50 0.72M ݸ, MPT0B640 0.12M̱ ú񸣺 ׹̷ Ȱ 6 ̻ ϴٰ ߴ. ƿ﷯ ó MPT0B640 ڷγ19 ׹̷ ȿ δٴ ̱ FDA ڷγ19 ߰ IND غ ߿ ִٰ .  
޵ ؼ (junsoo@mdtoday.co.kr)


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